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Kmtcqp 08tis 13 a prototype drug a is a

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KMTC/QP-08/TIS13. A prototype drug;
14. Drugs with high lipophillicity;
15. Chemical bonding affects drug action in the following ways, except;
16. The products of S-dealkylation area)Aldehydes and thiolsb)Aldehydes and sulfonesc)Alcohols and thiolsd)Aldehydes and thioethers
17. Which of the following is not a crucial requirement for a drug to act as an agonist?
18. Hydrogen bonding affects the activity of drug molecules in the following ways except:
19. The common structural feature between β-blockers and isoprenaline is:
Section B.20. List the desirable properties of a pro-drug (4 marks)21. Explain why it may be necessary to formulate drugs as pro-drugs with relevant examples(4 Marks)5
KMTC/QP-08/TIS22.a.The following structure is a 4- phenyl piperidine, explain the phamarcophores in itwhich enables it act like an opioid (4 Marks)

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Term
Spring
Professor
NoProfessor
Tags
Pharmacology, Morphine, Paracetamol, Cetirizine, DEPARTMENT OF PHARMACY

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